An edition of Constitutive activity in receptors and other proteins
(2010)
Constitutive activity in receptors and other proteins
by P. Michael Conn
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Constitutive activity in receptors and other proteins
2010, Elsevier/Academic
electronic resource /
in English
0123812976 9780123812971
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Book Details
Table of Contents
v. 484. Constitutive activity at the cannabinoid CB(1) receptor and behavioral responses
Detecting constitutive activity and protean agonism at cannabinoid-2 receptor
Modulation of the constitutive activity of the ghrelin receptor by use of pharmacological tools and mutagenesis
Assessment of constitutive activity and internalization of GPR54 (KISS1-R)
Assessment of constitutive activity in E-type prostanoid receptors
[Alpha](1D-adrenergic receptors constitutive activity and reduced expression at the plasma membrane
Constitutive activity of the histamine H(1) receptor
Constitutive activity of somatostatin receptor subtypes
Assessment of homologous internalization of constitutively active N111G mutant of AT(1) receptor
Methods to detect cell surface expression and constitutive activity of GPR6
[beta](3)-adrenoceptor agonists and (antagonists as) inverse agonists history, perspective, constitutive activity, and stereospecific binding
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Constitutive activity of the lutropin receptor and its allosteric modulation by receptor heterodimerization
Assessing constitutive activity of extracellular calcium-sensing receptors in vitro and in bone
Constitutive activity of neural melanocortin receptors
Measurement of constitutive activity of bmp type I receptors
Probing the constitutive activity among dopamine D1 and D5 receptors and their mutants
Identification of gain-of-function variants of the human prolactin receptor
Investigations of activated ACVR1/ALK2, a bone morphogenetic protein type i receptor, that causes fibrodysplasia ossificans progressiva
Identification and evaluation of constitutively active thyroid stimulating hormone receptor mutations
Assessment of constitutive activity of a G protein-coupled receptor, CPR2, in cryptococcus neoformans by heterologous and homologous methods
In vitro and in vivo assessment of mu opioid receptor constitutive activity
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Constitutively active [mu]-opioid receptors
Protein kinase CK2 is a constitutively active enzyme that promotes cell survival: Strategies to identify CK2 substrates and manipulate its activity in mammalian cells
Assessment of CK2 constitutive activity in cancer cells
Structural basis of the constitutive activity of protein kinase CK2
Measuring the constitutive activation of C-jun N-terminal kinase isoforms
Measurement of constitutive mapk and PI3K/AKT signaling activity in human cancer cell lines
Constitutive activity of GPR40/FFA1 intrinsic or assay dependent?
Constitutive activity of trp channels methods for measuring the activity and its outcome
Measurement of orexin (hypocretin) and substance P effects on constitutively active inward rectifier K(+) channels in brain neurons
Characterization of G protein-coupled receptor kinase 4 and measuring its constitutive activity in vivo
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Voltage-clamp-based methods for the detection of constitutively active acetylcholine-gated I(K, ACH) channels in the diseased heart
Assaying WAVE and WASH complex constitutive activities toward the Arp2/3 complex
Methods to assess the mechanism of protein function.
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V.485. Identification and characterization of steroidogenic factor-1 inverse agonists
Assessment of inverse agonism for the angiotensin II type 1 receptor
Measurement of inverse agonism in [beta]-adrenoceptors
Techniques for studying inverse agonist activity of antidepressants at recombinant nonedited 5-HT(C-INI) receptor and native neuronal 5-HT(2C) receptors
Differential inverse agonism at the human muscarinic M3 receptor
Ghrelin receptor: High constitutive activity and methods for developing inverse agonists
Constitutive activity and inverse agonism at the [alpha](A) and [alpha](B) adrenergic receptor subtypes
Measurement of inverse agonism of the cannabinoid receptors
Constitutively active thyrotropin and thyrotropin-releasing hormone receptors and their inverse agonists
Inverse agonists and antagonists of retinoid receptors
[gamma]-aminobutyric acid type A (GABA(A)) receptor subtype inverse agonists as therapeutic agents in cognition
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Assays for inverse agonists in the visual system
Receptor-driven identification of novel human a adenosine receptor antagonists as potential therapeutic agents
Inverse agonist activity of steroidogenic factor SF-1
Methods to measure G-protein-coupled receptor activity for the identification of inverse agonists
Use of pharmacoperones to reveal GPCR structural changes associated with constitutive activation and trafficking
Application of large-scale transient transfection to cell-based functional assays for ion channels and GPCRs
Quantification of RNA editing of the serotonin 2C receptor (5-HT(C)R) ex vivo
Strategies for isolating constitutively active and dominant-negative pheromone receptor mutants in yeast
Development of a GPR23 cell-based [beta]-lactamase reporter assay
Computational modeling of constitutively active mutants of GPCRs C5A receptor
TSH receptor monoclonal antibodies with agonist, antagonist, and inverse agonist activities
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Current standards, variations, and pitfalls for the determination of constitutive TSHR activity in vitro
Toward the rational design of constitutively active KCA3.1 mutant channels
Fusion proteins as model systems for the analysis of constitutive GPCR activity
Screening for novel constitutively active CXCR2 mutants and their cellular effects
A method for parallel solid-phase synthesis of iodinated analogs of the cannabinoid receptor type I (CB) inverse agonist rimonabant
Coexpression systems as models for the analysis of constitutive GPCR activity
Modeling and simulation of inverse agonism dynamics
Design and use of constitutively active STAT5 constructs
In vitro and in vivo assays of protein kinase CK2 activity.
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Edition Notes
Includes bibliographical references and indexes.
Description based on print version record.
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